SCHEMBL10103477

SCHEMBL10103477

Cc1nc(NCCc2ccccc2)sc1C(=O)N[C@H]1CCC2CC3C[C@@](O)(C2)CC31

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.52
HSD11B1 P28845 10/20 0.44
RAB9A P51151 3/20 0.41
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
SCD O00767 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10086121 0.86 HSD11B1 (0.61) NPC1HSD11B1
SCHEMBL525571 0.86 HSD11B1 (0.61) NPC1HSD11B1
SCHEMBL10103468 0.83 HIF1A (0.40) NPC1HSD11B1RAB9AALDH1A1SMN1; SMN2
SCHEMBL10103461 0.76 HTT (0.36) NPC1HSD11B1RAB9AALDH1A1SMN1; SMN2
SCHEMBL10103199 0.75 HTR3E (0.42) HSD11B1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL10103445 0.73 HSD11B1 (0.42) NPC1HSD11B1RAB9AALDH1A1SMN1; SMN2
SCHEMBL525062 0.70 NPC1 (1.00) NPC1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL14135317 0.69 FAAH (0.45) NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL10086305 0.69 HSD11B1 (0.52) HSD11B1
SCHEMBL525274 0.69 HSD11B1 (0.52) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012015715-A1 SUBSTITUTED THIAZOL-2-YLAMINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE AS 11-BETA HSD1 MODULATORS HIGH POINT PHARMACEUTICALS, LLC (US) 2012-02-02 WO disclosed