SCHEMBL10104355

SCHEMBL10104355

Cc1cc(NCCN(C)C)c(Cl)c(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
NCF1 P14598 2/20 0.36
CHEK1 O14757 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
RPS6KB1 P23443 1/20 0.35
AKT1 P31749 1/20 0.35
AKT2 P31751 1/20 0.35
RPS6KA3 P51812 1/20 0.35
BRD4 O60885 1/20 0.33
ATAD2 Q6PL18 1/20 0.33
UTS2R Q9UKP6 1/20 0.33
PTGES O14684 1/20 0.33
NOS2 P35228 2/20 0.33
ALPL P05186 1/20 0.33
ALPI P09923 1/20 0.33
NOS1 P29475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10104381 0.85 NCF1 (0.38) ALDH1A1NPSR1NCF1CHEK1MEN1
SCHEMBL10104393 0.84 NCF1 (0.37) ALDH1A1NPSR1NCF1CHEK1MEN1
SCHEMBL10104410 0.75 ACHE (0.40) MEN1KMT2APTGES
SCHEMBL10104319 0.73 RAPGEF4 (0.33) UTS2R
SCHEMBL15517270 0.71 RAPGEF4 (0.42) ALDH1A1MEN1KMT2A
SCHEMBL10104357 0.71 RAPGEF4 (0.32) NPSR1MEN1KMT2AUTS2RNOS2
SCHEMBL10104437 0.70 SLC6A4 (0.42) ALDH1A1L3MBTL1MEN1KMT2ANOS2
SCHEMBL10104260 0.69 RAPGEF4 (0.44) NOS2NOS1
SCHEMBL9023734 0.69 POLB (0.43) ALDH1A1NPSR1NCF1CHEK1MEN1
SCHEMBL10104369 0.68 NCF1 (0.38) ALDH1A1NPSR1NCF1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889665-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-18 US disclosed
US-8778929-B2 Substituted heteroaryl inhibitors of B-RAF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-07-15 US disclosed
US-8653087-B2 Pyrido [5, 4-D] pyrimidines as cell proliferation inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-02-18 US disclosed
US-20120094975-A1 PYRIDO [5, 4-D] PYRIMIDINES AS CELL PROLIFERATION INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-04-19 US disclosed
US-20110312939-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-12-22 US disclosed
US-20110183952-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183952-A1 NEW CHEMICAL COMPOUNDS MKI67, CCNA1, CCNT1 ALDH1A1 75/4885NPSR1 460/4885L3MBTL1 746/4885
US-20110312939-A1 NEW CHEMICAL COMPOUNDS CCNA1, CCNT1, MKI67 ALDH1A1 175/4885NPSR1 987/4885L3MBTL1 459/4885
US-20120094975-A1 PYRIDO [5, 4-D] PYRIMIDINES AS CELL PROLIFERATION INHIBITORS CCNT1, CCNA1, CCND1 ALDH1A1 860/4885NPSR1 1418/4885L3MBTL1 283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.