SCHEMBL10104358

SCHEMBL10104358

Cc1cc(OC(F)(F)F)cc(N2CCCN(C)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.47
ALDH1A1 P00352 1/20 0.43
CHKA P35790 1/20 0.41
MAP4K1 Q92918 1/20 0.40
CCR6 P51684 2/20 0.40
MCHR1 Q99705 1/20 0.40
DDR1 Q08345 1/20 0.40
NCF1 P14598 1/20 0.40
LMNA P02545 1/20 0.40
TRPV4 Q9HBA0 2/20 0.39
PHGDH O43175 1/20 0.39
HTR3A P46098 1/20 0.38
PDK2 Q15119 1/20 0.37
GRIN2B Q13224 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10104342 0.94 FFAR4 (0.51) FFAR4ALDH1A1MAP4K1CCR6DDR1
SCHEMBL10104356 0.79 TSHR (0.54) FFAR4ALDH1A1MCHR1DDR1PHGDH
SCHEMBL19457814 0.78 ADRB1 (0.53) FFAR4ALDH1A1DDR1HTR3A
SCHEMBL10104546 0.78 FFAR4 (0.50) FFAR4ALDH1A1DDR1LMNA
SCHEMBL10104302 0.78 ADRB1 (0.45) FFAR4ALDH1A1CHKANCF1LMNA
SCHEMBL10104531 0.77 FFAR4 (0.47) FFAR4ALDH1A1
SCHEMBL24123750 0.76 ADRB1 (0.51) FFAR4ALDH1A1PHGDHHTR3A
SCHEMBL2056171 0.76 ALDH1A1 (0.59) ALDH1A1MAP4K1LMNATRPV4HTR3A
SCHEMBL12968842 0.75 ADRA2C (0.56) ALDH1A1CCR6PHGDHHTR3A
SCHEMBL12359403 0.73 MAPT (0.54) ALDH1A1LMNAHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889665-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-18 US disclosed
US-8778929-B2 Substituted heteroaryl inhibitors of B-RAF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-07-15 US disclosed
US-8653087-B2 Pyrido [5, 4-D] pyrimidines as cell proliferation inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-02-18 US disclosed
US-20120094975-A1 PYRIDO [5, 4-D] PYRIMIDINES AS CELL PROLIFERATION INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-04-19 US disclosed
US-20110312939-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-12-22 US disclosed
US-20110183952-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183952-A1 NEW CHEMICAL COMPOUNDS MKI67, CCNA1, CCNT1 FFAR4 4456/4885ALDH1A1 75/4885CHKA 2333/4885
US-20110312939-A1 NEW CHEMICAL COMPOUNDS CCNA1, CCNT1, MKI67 FFAR4 4204/4885ALDH1A1 175/4885CHKA 2530/4885
US-20120094975-A1 PYRIDO [5, 4-D] PYRIMIDINES AS CELL PROLIFERATION INHIBITORS CCNT1, CCNA1, CCND1 FFAR4 2848/4885ALDH1A1 860/4885CHKA 3309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.