SCHEMBL10105030

SCHEMBL10105030

Cc1cn(C)c(=O)[nH]c1=S

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.39
TK1 P04183 1/20 0.34
P2RY2 P41231 1/20 0.33
DAO P14920 2/20 0.32
BRD4 O60885 1/20 0.31
LPO P22079 1/20 0.30
PTGS1 P23219 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
TSHR P16473 1/20 0.30
MAPK10 P53779 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18069601 0.77 ALDH1A1 (0.34) LPOPTGS1SMN1; SMN2
SCHEMBL16248 0.77 MAPK1 (0.47) CRBNTK1DAOMAPK1
SCHEMBL21836662 0.77 CRBN (0.38) CRBNP2RY2DAO
SCHEMBL16575631 0.77 CRBN (0.38) CRBNP2RY2DAO
SCHEMBL6420314 0.76 MAPK1 (0.46) CRBNTK1DAOMAPK1
SCHEMBL7546901 0.75 TK1 (0.42) TK1MAPK1
SCHEMBL20998663 0.74 CRBN (0.39) CRBNDAOBRD4SMN1; SMN2MAPK1
SCHEMBL22571159 0.74 ALDH1A1 (0.34) TK1
SCHEMBL11723021 0.74 SMN1; SMN2 (0.44) TK1LPOSMN1; SMN2MAPK1
SCHEMBL7554990 0.72 TK1 (0.47) TK1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3632468-B1 5-IODO-4-THIO-2'-DEOXYURIDINE FOR USE AS A RADIOSENSITIZER IN RADIOTHERAPY UNIV GDANSKI (PL) 2023-12-13 EP disclosed
US-9732110-B2 Nucleoside and nucleotide derivatives ENANTA PHARMACEUTICALS, INC. (US) 2017-08-15 US disclosed
US-8163707-B2 4′-allene-substituted nucleoside derivatives ENANTA PHARMACEUTICALS, INC. (US) 2012-04-24 US disclosed
US-20100074889-A1 4'-ALLENE-SUBSTITUTED NUCLEOSIDE DERIVATIVES ENANTA PHARMACEUTICALS, INC. 2010-03-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100074889-A1 4'-ALLENE-SUBSTITUTED NUCLEOSIDE DERIVATIVES CCNI, CCNA1, CDK1 CRBN 4591/4885TK1 29/4885P2RY2 2338/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.