SCHEMBL7546901

SCHEMBL7546901

CCCn1cc(C)c(=S)[nH]c1=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TK1 P04183 3/20 0.42
TYMP P19971 1/20 0.40
MAPK1 P28482 1/20 0.39
HPGD P15428 1/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2C19 P33261 3/20 0.38
GAA P10253 1/20 0.38
MEN1 O00255 1/20 0.38
CYP2C9 P11712 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TYR P14679 1/20 0.38
LMNA P02545 1/20 0.37
TK2 O00142 4/20 0.37
PDE4A P27815 1/20 0.36
ADORA2A P29274 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7554990 0.90 TK1 (0.47) TK1TYMPMAPK1HPGDCYP1A2
SCHEMBL11723021 0.85 SMN1; SMN2 (0.44) TK1TYMPMAPK1HPGD
SCHEMBL4118603 0.81 MAPK1 (0.57) TK1TYMPMAPK1HPGDTK2
SCHEMBL28985700 0.79 LMNA (0.42) TK1TYMPMAPK1GAACYP2C9
SCHEMBL7549198 0.77 TYMP (0.43) TK1TYMPMAPK1HPGD
SCHEMBL10105030 0.75 CRBN (0.39) TK1MAPK1
SCHEMBL28985696 0.75 TK1 (0.37) TK1TYMPMAPK1HPGDKMT2A
SCHEMBL7546248 0.73 HPGD (0.72) TK1MAPK1HPGD
SCHEMBL7679806 0.70 CYP2C19 (0.40) TYMPHPGDCYP1A2CYP2C19GAA
SCHEMBL13261412 0.70 TK1 (0.62) TK1TYMPMAPK1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165554-A1 NEW ENDOTHELIN CONVERTING ENZYME INHIBITORS, THEIR PRODUCTION AND THEIR USE BASF AKTIENGESELLSCHAFT (DE) 2002-01-02 EP disclosed
WO-2000061579-A1 NEW ENDOTHELIN CONVERTING ENZYME INHIBITORS, THEIR PRODUCTION AND THEIR USE BASF AKTIENGESELLSCHAFT (DE) 2000-10-19 WO disclosed