SCHEMBL1011623

SCHEMBL1011623

Fc1ccc(Oc2cccc(C=C3CCNCC3)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.43
SLC6A4 P31645 8/20 0.43
SLC6A3 Q01959 7/20 0.43
HTR1A P08908 6/20 0.43
AKR1B1 P15121 1/20 0.41
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
ALOX12 P18054 1/20 0.40
NFKB1 P19838 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1011388 0.99 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3HTR1AAKR1B1
SCHEMBL1009494 0.88 AKR1B1 (0.51) AKR1B1MAPTMEN1KMT2ALMNA
SCHEMBL1013799 0.86 LTA4H (0.42) AKR1B1MEN1KMT2AALOX5ADAMTS5
Hydrochloric Acid SCHEMBL1010352 0.84 ADAMTS5 (0.55) ADAMTS5
SCHEMBL1011559 0.83 ADAMTS5 (0.43) AKR1B1ADAMTS5MMP3MMP13
SCHEMBL27233690 0.82 FAAH (0.46) CYP3A4CYP2D6CYP2C9
SCHEMBL27233592 0.79 RAB9A (0.43) AKR1B1MAPTALDH1A1LMNAALOX5
SCHEMBL28683291 0.79 IKBKB (0.54) CYP1A2CYP3A4CYP2D6MAPK1BLM
SCHEMBL27763712 0.78 ELANE (0.50) AKR1B1MEN1ALDH1A1KMT2ALMNA
SCHEMBL27233568 0.78 HTR2C (0.50) AKR1B1MAPTMEN1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076508-B1 BIARYL ETHER UREA COMPOUNDS PFIZER PROD INC (US) 2011-01-05 EP disclosed
EP-2076508-A2 BIARYL ETHER UREA COMPOUNDS Pfizer Products Inc. (US) 2009-07-08 EP disclosed
WO-2008047229-A2 BIARYL ETHER UREA COMPOUNDS PFIZER PRODUCTS INC. (US) 2008-04-24 WO disclosed