SCHEMBL10117698

SCHEMBL10117698

CCOC(=O)N(C(=O)OCC)c1ncc(-c2ccc(Br)cc2)n1C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.41
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
NR1H2 P55055 7/20 0.36
HTT P42858 1/20 0.36
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
TARBP2 Q15633 1/20 0.34
MAPT P10636 4/20 0.33
NR1H3 Q13133 3/20 0.33
GPR119 Q8TDV5 1/20 0.33
POLB P06746 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KCNK3 O14649 1/20 0.33
KCNK9 Q9NPC2 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
CHRNA7 P36544 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10117696 0.92 NR1H2 (0.37) IDO1MEN1NPC1RAB9AKMT2A
SCHEMBL10117875 0.88 NPC1 (0.35) IDO1MEN1NPC1RAB9AKMT2A
SCHEMBL24176651 0.79 NR1H2 (0.38) NR1H2NR1H3GPR119AAK1
SCHEMBL10117534 0.76 NR1H2 (0.40) IDO1MEN1KMT2ANR1H2MAPT
SCHEMBL13655217 0.74 NR1H2 (0.35) NR1H2NR1H3GPR119AAK1
SCHEMBL10117536 0.73 MTOR (0.38) IDO1MEN1KMT2ANR1H2
SCHEMBL13663132 0.72 PTPN1 (0.53) MEN1NPC1RAB9AKMT2AMAPT
SCHEMBL13655220 0.72 HDAC8 (0.43) MEN1KMT2ANR1H2MAPTAAK1
SCHEMBL10117508 0.72 NPC1 (0.41) IDO1MEN1NPC1RAB9AKMT2A
SCHEMBL24176646 0.72 HDAC2 (0.35) NPC1RAB9ANR1H2NR1H3GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087976-A2 NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-06-28 WO disclosed