SCHEMBL10117696

SCHEMBL10117696

CCCOC(=O)N(C(=O)OCCC)c1ncc(-c2ccc(Br)cc2)n1C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 8/20 0.37
IDO1 P14902 1/20 0.36
NR1H3 Q13133 3/20 0.33
GABRA2 P47869 1/20 0.32
GABRB2 P47870 1/20 0.32
HRH2 P25021 1/20 0.32
HRH1 P35367 1/20 0.32
KCNK3 O14649 3/20 0.32
KCNK9 Q9NPC2 3/20 0.32
AAK1 Q2M2I8 1/20 0.32
THRB P10828 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
BCL2 P10415 1/20 0.31
BECN1 Q14457 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10117698 0.92 IDO1 (0.41) NR1H2IDO1NR1H3HRH2HRH1
SCHEMBL10117875 0.86 NPC1 (0.35) NR1H2IDO1NR1H3AAK1MEN1
SCHEMBL24176651 0.77 NR1H2 (0.38) NR1H2NR1H3AAK1
SCHEMBL13655217 0.74 NR1H2 (0.35) NR1H2NR1H3GABRA2AAK1
SCHEMBL10117534 0.74 NR1H2 (0.40) NR1H2IDO1NR1H3KCNK3KCNK9
SCHEMBL10117508 0.72 NPC1 (0.41) NR1H2IDO1MEN1NPC1RAB9A
SCHEMBL10117536 0.72 MTOR (0.38) NR1H2IDO1MEN1KMT2ABCL2
SCHEMBL13663132 0.71 PTPN1 (0.53) MEN1NPC1RAB9AKMT2A
SCHEMBL10117537 0.71 RAB9A (0.49) NR1H2IDO1NPC1RAB9A
SCHEMBL13655220 0.71 HDAC8 (0.43) NR1H2AAK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087976-A2 NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-06-28 WO disclosed