SCHEMBL10119795

SCHEMBL10119795

CCCn1cc(CCNC)c2ccc(OC)cc21

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.56
HTR2A P28223 1/20 0.46
MTNR1A P48039 3/20 0.44
MTNR1B P49286 3/20 0.44
NQO2 P16083 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
DYRK1A Q13627 1/20 0.42
ADRB2 P07550 2/20 0.41
CNR2 P34972 1/20 0.41
HASPIN Q8TF76 1/20 0.41
SSTR5 P35346 1/20 0.41
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
NR1D1 P20393 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25418921 0.90 HTR6 (0.70) HTR6HTR2AMTNR1AMTNR1BNQO2
SCHEMBL8271864 0.88 HTR6 (0.62) HTR6MTNR1AMTNR1BNQO2HDAC3
SCHEMBL8270015 0.84 ADRB2 (0.59) HTR6HTR2ADYRK1AADRB2CNR2
SCHEMBL9883700 0.79 HTR6 (0.45) HTR6HTR2AMTNR1AMTNR1BNQO2
SCHEMBL19650681 0.78 HTR6 (0.52) HTR6CNR2NR1D1
SCHEMBL8271739 0.76 ALDH1A1 (0.52) HTR6CNR2SSTR5MEN1KMT2A
SCHEMBL24878072 0.75 HTR6 (0.57) HTR6HTR2AMTNR1AMTNR1BNQO2
SCHEMBL984866 0.72 L3MBTL1 (0.47) HTR6DYRK1ACNR2MEN1KMT2A
SCHEMBL25623396 0.71 HTR6 (0.81) HTR6HTR2A
SCHEMBL12641863 0.70 HTR6 (0.51) HTR6SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781639-B1 SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE JANSSEN PHARMACEUTICA NV (BE) 2012-01-25 EP disclosed