SCHEMBL10123931

SCHEMBL10123931

CCN1CCC(=C2c3ccc(Cl)cc3CCc3cccnc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 17/20 1.00
FNTA P49354 1/20 0.75
FNTB P49356 1/20 0.75
PTAFR P25105 2/20 0.72
SLC6A15 Q9H2J7 1/20 0.72
KCNH2 Q12809 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20952209 0.89 HRH1 (0.80) HRH1FNTAFNTBPTAFRSLC6A15
SCHEMBL20951899 0.88 HRH1 (0.79) HRH1FNTAFNTBPTAFRSLC6A15
SCHEMBL31384618 0.88 HRH1 (0.82) HRH1FNTAFNTBPTAFRSLC6A15
SCHEMBL29626502 0.88 HRH1 (0.82) HRH1FNTAFNTBPTAFRSLC6A15
SCHEMBL4460572 0.88 HRH1 (0.82) HRH1FNTAFNTBPTAFRSLC6A15
SCHEMBL20951362 0.87 HRH1 (0.77) HRH1FNTAFNTBPTAFRSLC6A15
SCHEMBL29279006 0.87 HRH1 (0.77) HRH1FNTAFNTBPTAFRSLC6A15
SCHEMBL8580306 0.87 HRH1 (0.77) HRH1FNTAFNTBPTAFRSLC6A15
SCHEMBL9139059 0.86 HRH1 (1.00) HRH1FNTAFNTBPTAFRKCNH2
SCHEMBL9136454 0.86 HRH1 (1.00) HRH1FNTAFNTBPTAFRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230140276-A1 TRICYCLIC COMPOUNDS, PREPARATION METHOD AND MEDICAL USE THEREOF HEFEI AMVITE PHARMACEUTICAL CO., LTD. (CN) 2023-05-04 US disclosed
EP-3319987-B1 NOVEL P450-BM3 VARIANTS WITH IMPROVED ACTIVITY CODEXIS INC (US) 2021-05-05 EP disclosed
US-8101782-B2 Drug hybrid of rivastigmine or physostigmine with tranylcypromine, amoxapine, desipramine, nortriptyline, protriptyline, fluoxetine, fluvoxamine, paroxetine, duloxetine, betahistine, amlodipine, proylhexedrine, rimantadine, desloratadine; Alzheimer's disease; Parkinson's disease, impairment in memory COLUCID PHARMACEUTICALS, INC. (US) 2012-01-24 US disclosed
US-20080261950-A1 Compounds that inhibit cholinesterase COLUCID PHARMACEUTICALS, INC. (US) 2008-10-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230140276-A1 TRICYCLIC COMPOUNDS, PREPARATION METHOD AND MEDICAL USE THEREOF HNMT, CHRM1, HRH4 HRH1 6/4885FNTA 2436/4885FNTB 3622/4885
US-20080261950-A1 Compounds that inhibit cholinesterase ACHE, BCHE, CHAT HRH1 765/4885FNTA 718/4885FNTB 1781/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.