SCHEMBL10129614

SCHEMBL10129614

CCOC(=O)c1ccc(Cl)nc1N[C@H]1CCCC[C@@H]1N1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR2F2 P24468 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MAPK1 P28482 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
SIGMAR1 Q99720 2/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
S1PR2 O95136 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
XBP1 P17861 1/20 0.39
PPP1CA P62136 1/20 0.39
OPRK1 P41145 6/20 0.39
SYK P43405 1/20 0.39
OPRM1 P35372 1/20 0.38
CHRNA7 P36544 1/20 0.38
DYRK1A Q13627 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10129609 0.84 FER (0.45) NR2F2NPSR1MAPK1KDM4EMAPT
SCHEMBL496019 0.81 NR2F2 (0.53) NR2F2NPSR1MAPK1KDM4EMAPT
SCHEMBL496058 0.76 ALOX15 (0.45) MAPK1KDM4ESIGMAR1KMT2AALDH1A1
SCHEMBL495858 0.76 MAPK1 (0.44) MAPK1KDM4EMAPTSIGMAR1KMT2A
SCHEMBL496781 0.73 PTGER4 (0.49) NPSR1RAB9AKMT2AMEN1DYRK1A
SCHEMBL495986 0.73 SMN1; SMN2 (0.56) MAPK1MAPTSIGMAR1KMT2AMEN1
SCHEMBL20891573 0.72 KDM4E (0.48) KDM4EMAPTNPC1RAB9AKMT2A
SCHEMBL20891566 0.70 TSHR (0.41) NPSR1KDM4EMAPTRAB9AKMT2A
SCHEMBL22860320 0.70 RIPK1 (0.47) KDM4EALDH1A1OPRK1SYK
SCHEMBL12936321 0.69 RIPK1 (0.49) KDM4EALDH1A1OPRK1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106190-B2 2-aminobenzamide derivatives ASTELLAS PHARMA INC. (JP) 2012-01-31 US disclosed
US-8106190-B2 2-aminobenzamide derivatives ASTELLAS PHARMA INC. (JP) 2012-01-31 US disclosed
US-20090233900-A1 2-AMINOBENZAMIDE DERIVATIVE ASTELLAS PHARMA INC. (JP) 2009-09-17 US disclosed
US-20090233900-A1 2-AMINOBENZAMIDE DERIVATIVE ASTELLAS PHARMA INC. (JP) 2009-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233900-A1 2-AMINOBENZAMIDE DERIVATIVE TRPV1, TRPV2, TRPV5 NR2F2 2185/4885NPSR1 513/4885MAPK1 1633/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.