SCHEMBL1014016

SCHEMBL1014016

CN(CC(C)(NC(=O)OC(C)(C)C)c1cc(F)cc(F)c1)C1(C(=O)O)CCCCC1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSD P07339 10/20 0.35
BACE1 P56817 10/20 0.35
RIPK1 Q13546 2/20 0.32
RORC P51449 1/20 0.32
DPP8 Q6V1X1 1/20 0.30
DPP9 Q86TI2 1/20 0.30
AAK1 Q2M2I8 1/20 0.30
FAAH O00519 1/20 0.30
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1013637 0.78 RIPK1 (0.34) CTSDBACE1RIPK1
SCHEMBL1012605 0.77 RIPK1 (0.34) CTSDBACE1RIPK1
SCHEMBL977080 0.74 BACE1 (0.35) CTSDBACE1RORCDPP8DPP9
SCHEMBL979457 0.73 BACE1 (0.33) CTSDBACE1RORCDPP8DPP9
SCHEMBL3695612 0.70 CTSS (0.34) AAK1
SCHEMBL17040319 0.68 APLNR (0.38) AAK1
SCHEMBL980274 0.67 CTSS (0.39) AAK1
SCHEMBL1225573 0.67 DRD2 (0.36) RIPK1
SCHEMBL16704779 0.66 CYP2C19 (0.31)
SCHEMBL6343801 0.65 AAK1 (0.36) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271346-A2 MONOCYCLIC CGRP RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2011-01-12 EP disclosed
WO-2009120652-A2 MONOCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2009-10-01 WO disclosed