SCHEMBL10146209

SCHEMBL10146209

CC(C)C1CCC(=O)CN1C

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.38
PIK3CD O00329 1/20 0.31
TOP2A P11388 1/20 0.30
TOP2B Q02880 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2757452 0.78 MAPK1 (0.35) MAPK1PIK3CDTOP2ATOP2BALDH1A1
SCHEMBL6628720 0.71
SCHEMBL27326433 0.70 SRD5A1 (0.39) MAPK1PIK3CD
SCHEMBL9980265 0.70 SRD5A1 (0.39) MAPK1PIK3CD
SCHEMBL10303898 0.70 SRD5A1 (0.39) MAPK1PIK3CD
SCHEMBL26546891 0.69 PIK3C3 (0.35) PIK3CDTOP2ATOP2BALDH1A1MAPT
SCHEMBL29180235 0.67 MAPK1 (0.33) MAPK1
SCHEMBL7600246 0.67 PIK3CD (0.36) PIK3CD
SCHEMBL6788884 0.67 MAPK1 (0.33) MAPK1
SCHEMBL29180234 0.67 MAPK1 (0.33) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-8999967-B2 Tricyclic fused ring inhibitors of hepatitis C PRESIDIO PHARMACEUTICALS, INC. (US) 2015-04-07 US disclosed
US-20130296304-A1 TRICYCLIC FUSED RING INHIBITORS OF HEPATITIS C PRESIDIO PHARMACEUTICALS, INC. (US) 2013-11-07 US disclosed
US-20120115855-A1 INHIBITORS OF HCV NS5A PRESIDIO PHARMACEUTICALS, INC. (US) 2012-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230133132-A1 NAMPT MODULATORS NAMPT, MC4R, SIRT1 MAPK1 846/4885PIK3CD 3016/4885TOP2A 4766/4885
US-20130296304-A1 TRICYCLIC FUSED RING INHIBITORS OF HEPATITIS C HAVCR2, HCCS, LIPC MAPK1 4154/4885PIK3CD 615/4885TOP2A 694/4885
US-20120115855-A1 INHIBITORS OF HCV NS5A HAVCR2, MAVS, EIF2AK2 MAPK1 2629/4885PIK3CD 391/4885TOP2A 2754/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.