SCHEMBL10147500

SCHEMBL10147500

CC(C)(Sc1ccc(Cl)cc1)C(=O)NN

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.43
KDM4E B2RXH2 5/20 0.43
MAPT P10636 5/20 0.43
LMNA P02545 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP2C19 P33261 3/20 0.37
CYP2C9 P11712 2/20 0.37
HSD17B10 Q99714 1/20 0.37
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 2/20 0.36
HSP90AA1 P07900 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10147498 0.83 ALDH1A1 (0.42) ALDH1A1KDM4EMAPTLMNAL3MBTL1
SCHEMBL4398676 0.78 PPARA (0.51) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL11539611 0.74 SLC22A12 (0.48) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL10999042 0.73 TBXAS1 (0.38) ALDH1A1MAPTLMNAL3MBTL1MEN1
SCHEMBL3323151 0.73 FFAR2 (0.52) ALDH1A1KDM4EMAPTLMNAL3MBTL1
SCHEMBL8418761 0.70 POLB (0.39) KDM4EMAPTLMNAPDK1PDK2
SCHEMBL11870199 0.70 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTLMNAL3MBTL1
SCHEMBL469433 0.70 CYP1A2 (0.56) ALDH1A1MAPTL3MBTL1POLBTDP1
SCHEMBL11538993 0.70 PPARA (0.51) ALDH1A1MAPTMEN1KMT2ACYP2C19
SCHEMBL11303469 0.69 MAPT (0.38) ALDH1A1MAPTLMNAL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418207-A1 Sulfone compounds which modulate the CB2 receptor Boehringer Ingelheim International GmbH (DE) 2012-02-15 EP disclosed