SCHEMBL10153310

SCHEMBL10153310

COC(=O)c1cc(Br)ccc1C(C(=O)OC)C(=O)OC

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.47
ALDH1A1 P00352 2/20 0.46
GAA P10253 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.43
HSD17B10 Q99714 1/20 0.43
SLC6A3 Q01959 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
HPGD P15428 3/20 0.41
CHEK1 O14757 1/20 0.39
TSHR P16473 2/20 0.39
HTT P42858 1/20 0.39
MAPT P10636 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15766202 0.86 NR4A2 (0.46) NR4A2ALDH1A1GAAL3MBTL1HSD17B10
SCHEMBL4084280 0.83 NR4A2 (0.53) NR4A2ALDH1A1GAAL3MBTL1HSD17B10
SCHEMBL30058887 0.83 NR4A2 (0.53) NR4A2ALDH1A1GAAL3MBTL1HSD17B10
SCHEMBL16034830 0.82 NR4A2 (0.48) NR4A2ALDH1A1GAAL3MBTL1HSD17B10
SCHEMBL10154075 0.81 SLC6A4 (0.43) ALDH1A1SLC6A3SMN1; SMN2HPGDTSHR
SCHEMBL10153655 0.81 ABL1 (0.53) NR4A2ALDH1A1SLC6A3SMN1; SMN2CHEK1
SCHEMBL18525601 0.78 HSD17B10 (0.44) NR4A2ALDH1A1GAAL3MBTL1HSD17B10
SCHEMBL22667294 0.77 ALDH1A1 (0.39) NR4A2ALDH1A1GAAL3MBTL1MAPT
SCHEMBL9961071 0.77 SMN1; SMN2 (0.57) ALDH1A1HSD17B10SMN1; SMN2HPGDHTT
SCHEMBL4577829 0.77 NR4A2 (0.56) NR4A2ALDH1A1GAAL3MBTL1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed