SCHEMBL10153655

SCHEMBL10153655

COC(=O)c1cc(Cl)ccc1C(C(=O)OC)C(=O)OC

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.53
NR4A2 P43354 2/20 0.47
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
RXFP1 Q9HBX9 1/20 0.43
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
LMNA P02545 4/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ALPL P05186 1/20 0.40
CHEK1 O14757 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15766246 0.84 ABL1 (0.50) ABL1NR4A2SLC6A4SLC6A3RXFP1
SCHEMBL3533537 0.81 LMNA (0.47) MEN1KMT2ALMNAALDH1A1NPC1
SCHEMBL4278397 0.81 ABL1 (0.53) ABL1NR4A2SLC6A4SLC6A3RXFP1
SCHEMBL10153310 0.81 NR4A2 (0.47) NR4A2SLC6A3ALDH1A1SMN1; SMN2MAPT
SCHEMBL10154075 0.81 SLC6A4 (0.43) SLC6A4SLC6A3ALDH1A1KDM4ENPC1
SCHEMBL10153993 0.79 NPC1 (0.50) ABL1SLC6A4SLC6A3ALDH1A1KDM4E
SCHEMBL15075786 0.79 ABL1 (0.54) ABL1MEN1KMT2ALMNAALDH1A1
SCHEMBL2535669 0.78 ABL1 (0.54) ABL1NR4A2SLC6A4SLC6A3RXFP1
SCHEMBL4234236 0.77 SMN1; SMN2 (0.49) ABL1MEN1KMT2AALDH1A1KDM4E
SCHEMBL9961071 0.77 SMN1; SMN2 (0.57) MEN1KMT2ALMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed