SCHEMBL10153993

SCHEMBL10153993

COC(=O)c1cc(Cl)ccc1C(C(=O)NOCc1ccccc1)C(=O)OC

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
CNR1 P21554 1/20 0.43
PLA2G2A P14555 1/20 0.42
PYGL P06737 1/20 0.41
ABL1 P00519 1/20 0.40
NOS2 P35228 1/20 0.40
PSMB5 P28074 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CASP3 P42574 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
SLC7A5 Q01650 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10154006 0.88 NPC1 (0.39) NPC1RAB9AKDM4EALDH1A1GAA
SCHEMBL10153733 0.87 NPC1 (0.49) NPC1RAB9APLA2G2AALDH1A1
SCHEMBL10153651 0.87 PLA2G2A (0.42) NPC1RAB9APLA2G2ANOS2PSMB5
SCHEMBL10153986 0.83 RAB9A (0.49) NPC1RAB9AALDH1A1GAA
SCHEMBL10153984 0.83 SMN1; SMN2 (0.47) NPC1RAB9AKDM4EGAA
SCHEMBL10153654 0.81 NPC1 (0.47) NPC1RAB9AALDH1A1GAASLC7A5
SCHEMBL10153987 0.81 NPC1 (0.44) NPC1RAB9AKDM4E
SCHEMBL10153655 0.79 ABL1 (0.53) NPC1RAB9AABL1SLC6A4SLC6A3
SCHEMBL9789583 0.71 PTGER1 (0.61) CNR1
SCHEMBL1095126 0.71 CASP3 (0.58) NPC1RAB9ACNR1PLA2G2ACASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed