SCHEMBL10153683

SCHEMBL10153683

COC(=O)c1cc(NC(=O)c2ccccn2)ccc1C(C(=O)OC)C(=O)OC

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.56
NPC1 O15118 5/20 0.56
RAB9A P51151 5/20 0.56
KDM4E B2RXH2 2/20 0.56
GRM4 Q14833 15/20 0.54
HDAC6 Q9UBN7 1/20 0.54
PKM P14618 2/20 0.53
MAPT P10636 2/20 0.53
MITF O75030 1/20 0.51
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10153987 0.86 NPC1 (0.44) SMN1; SMN2NPC1RAB9AKDM4EGRM4
SCHEMBL10153281 0.83 SMN1; SMN2 (0.59) SMN1; SMN2NPC1RAB9AKDM4EMAPT
SCHEMBL9961071 0.79 SMN1; SMN2 (0.57) SMN1; SMN2NPC1RAB9AKDM4EPKM
SCHEMBL1657250 0.78 GRM4 (0.67) SMN1; SMN2NPC1RAB9AKDM4EGRM4
SCHEMBL4311315 0.74 SMN1; SMN2 (0.71) SMN1; SMN2NPC1RAB9AKDM4EGRM4
SCHEMBL11446166 0.72 POLB (0.60) SMN1; SMN2NPC1RAB9AKDM4EHDAC6
SCHEMBL10153655 0.71 ABL1 (0.53) SMN1; SMN2NPC1RAB9AKDM4EMAPT
SCHEMBL10153648 0.71 ALDH1A1 (0.59) SMN1; SMN2NPC1RAB9AKDM4EMAPT
SCHEMBL7990375 0.70 KDR (0.84) SMN1; SMN2NPC1RAB9AKDM4EGRM4
SCHEMBL23705777 0.70 GRM4 (1.00) SMN1; SMN2NPC1RAB9AKDM4EGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed