SCHEMBL10154006

SCHEMBL10154006

Bc1ccc(C(C(=O)NOCc2ccccc2)C(=O)OC)c(C(=O)OC)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
SLC7A5 Q01650 1/20 0.39
THRB P10828 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B10 Q99714 1/20 0.38
LTA4H P09960 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10153733 0.88 NPC1 (0.49) NPC1RAB9AALDH1A1LTA4HALOX15
SCHEMBL10153993 0.88 NPC1 (0.50) NPC1RAB9AALDH1A1KDM4EGAA
SCHEMBL10153651 0.88 PLA2G2A (0.42) NPC1RAB9AALDH1A1KDM4EGAA
SCHEMBL10153986 0.84 RAB9A (0.49) NPC1RAB9AALDH1A1GAALMNA
SCHEMBL10153984 0.83 SMN1; SMN2 (0.47) NPC1RAB9AKDM4EGAALMNA
SCHEMBL10153654 0.82 NPC1 (0.47) NPC1RAB9AALDH1A1GAASLC7A5
SCHEMBL10153987 0.80 NPC1 (0.44) NPC1RAB9AKDM4E
SCHEMBL10797269 0.68 LTA4H (0.51) NPC1RAB9AALDH1A1THRBCYP2C9
SCHEMBL21045042 0.68 RAB9A (0.39) NPC1RAB9AALDH1A1KDM4EHPGD
SCHEMBL10790971 0.67 LTA4H (0.53) NPC1RAB9AALDH1A1THRBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed