SCHEMBL1015454

SCHEMBL1015454

COC(=O)c1cc(Cl)ccc1NC(=O)COCC(=O)Nc1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPT P10636 4/20 0.46
KLK7 P49862 1/20 0.46
CETP P11597 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
P2RX1 P51575 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1015837 0.91 CNR1 (0.51) ALDH1A1KDM4EGAASMN1; SMN2MAPT
SCHEMBL1797516 0.90 ALDH1A1 (0.50) ALDH1A1KDM4EGAASMN1; SMN2MAPT
SCHEMBL1015269 0.89 GRIK1 (0.52) RAB9AKDM4EGAASMN1; SMN2MAPT
SCHEMBL1015634 0.89 ALDH1A1 (0.53) ALDH1A1KDM4EGAASMN1; SMN2MAPT
SCHEMBL1014545 0.88 KDM4E (0.46) ALDH1A1KDM4EGAASMN1; SMN2MAPT
SCHEMBL1015135 0.88 GRIK1 (0.51) RAB9AKDM4EGAASMN1; SMN2MAPT
SCHEMBL1015136 0.87 SLC6A4 (0.51) ALDH1A1KDM4EGAASMN1; SMN2MAPT
SCHEMBL1015137 0.87 KLK7 (0.46) ALDH1A1RAB9AGAASMN1; SMN2MAPT
SCHEMBL1013909 0.85 SERPINE1 (0.57) ALDH1A1KDM4EGAASMN1; SMN2MAPT
SCHEMBL1798637 0.85 KDM4E (0.52) ALDH1A1RAB9AKDM4EGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8415479-B2 Inhibitor of plasminogen activator inhibitor-1 RENASCIENCE CO., LTD. (JP) 2013-04-09 US disclosed
US-20110112140-A1 INHIBITOR OF PLASMINOGEN ACTIVATOR INHIBITOR-1 RENASCIENCE CO., LTD. (JP) 2011-05-12 US disclosed
EP-2272822-A1 INHIBITOR OF PLASMINOGEN ACTIVATOR INHIBITOR-1 Renascience CO., LTD. (JP) 2011-01-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110112140-A1 INHIBITOR OF PLASMINOGEN ACTIVATOR INHIBITOR-1 SERPINE1, SERPINB1, SERPINC1 ALDH1A1 888/4885RAB9A 2950/4885KDM4E 4108/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.