SCHEMBL10157089

SCHEMBL10157089

Cc1cc(CN(C(=O)OCc2ccccc2)c2ccccc2)ccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSPO P30536 2/20 0.42
ALDH1A1 P00352 3/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
PDK1 Q15118 2/20 0.41
KDM5A P29375 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
CHRM2 P08172 6/20 0.40
CHRM1 P11229 6/20 0.40
CHRM3 P20309 6/20 0.40
CHRM5 P08912 1/20 0.39
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
NPC1 O15118 1/20 0.39
GLA P06280 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
PAX8 Q06710 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PTGES O14684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10157569 0.85 GABRP (0.46) TSPOALDH1A1MAPTHPGDPDK1
SCHEMBL25920400 0.82 RAB9A (0.53) TSPOALDH1A1MAPTHPGDCHRM2
SCHEMBL3336342 0.82 GAA (0.50) ALDH1A1MAPTHPGDPDK1CHRM2
SCHEMBL10157007 0.80 TSHR (0.40) TSPOALDH1A1MAPTHPGDPDK1
SCHEMBL25920677 0.79 CNR2 (0.52) TSPOALDH1A1MAPTHPGDCHRM2
SCHEMBL14944354 0.79 JMJD6 (0.41) TSPOALDH1A1MAPTHPGDPDK1
SCHEMBL25920399 0.77 CHRM2 (0.43) ALDH1A1MAPTHPGDPDK1CHRM2
SCHEMBL3084308 0.74 ALDH1A1 (0.50) ALDH1A1MAPTHPGDCHRM2CHRM1
SCHEMBL19512871 0.74 RAB9A (0.48) TSPOALDH1A1MAPTGAANPC1
SCHEMBL3331879 0.74 GAA (0.61) ALDH1A1MAPTPDK1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052390-A1 N-2-(2-PYRIDINYL)-4-PYRIMIDINYL-BETA-ALANINE DERIVATIVES AS INHIBITORS OF HISTONE DEMETHYLASE JMJD3 GLAXO GROUP LIMITED (GB) 2012-04-26 WO disclosed