SCHEMBL10168025

SCHEMBL10168025

O=C(CNC(=O)c1cccnc1)c1ccc(Cl)c(O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.56
NPC1 O15118 4/20 0.51
RAB9A P51151 3/20 0.51
TSHR P16473 1/20 0.51
ALDH1A1 P00352 4/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
AGTR1 P30556 1/20 0.50
CYP2C19 P33261 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
KCNMA1 Q12791 1/20 0.49
ROCK2 O75116 1/20 0.48
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14212112 0.90 ALDH1A1 (0.62) THRBNPC1RAB9ATSHRALDH1A1
SCHEMBL23014252 0.80 TSHR (0.64) THRBNPC1RAB9ATSHRALDH1A1
SCHEMBL21391314 0.78 THRB (0.63) THRBNPC1RAB9ATSHRCYP1A2
SCHEMBL2817973 0.75 THRB (0.59) THRBRAB9AALDH1A1KMT2AGAA
SCHEMBL21378834 0.73 MAPT (0.65) THRBALDH1A1CYP2C9CYP2C19MEN1
SCHEMBL3864600 0.73 THRB (0.75) THRBNPC1RAB9ATSHRCYP1A2
Nicotinuric Acid SCHEMBL30183567 0.73 THRB (0.75) THRBNPC1RAB9ATSHRALDH1A1
Nicotinuric Acid SCHEMBL351962 0.73 THRB (0.75) THRBNPC1RAB9ATSHRALDH1A1
N-Hydroxymethylnicotinamide SCHEMBL352358 0.73 THRB (1.00) THRBNPC1RAB9ATSHRALDH1A1
SCHEMBL4869581 0.72 THRB (0.68) THRBNPC1RAB9ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534680-B1 PRENYLATION INHIBITORS AND METHODS OF THEIR SYNTHESIS AND USE PHARMACO INVESTMENTS INC (US) 2012-02-22 EP disclosed