SCHEMBL10169398

SCHEMBL10169398

CC(C)c1cccc(N(C)S(=O)(=O)c2cccnc2)c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
GRM2 Q14416 3/20 0.43
HSD17B1 P14061 3/20 0.43
HSD17B2 P37059 3/20 0.43
NAMPT P43490 1/20 0.41
F2 P00734 2/20 0.41
NAPRT Q6XQN6 1/20 0.40
NR1H3 Q13133 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10169327 0.83 NR1H3 (0.53) HSD17B1HSD17B2F2NR1H3L3MBTL1
SCHEMBL10211749 0.82 ALDH1A1 (0.52) CYP11B1CYP11B2HSD17B1HSD17B2F2
SCHEMBL9959448 0.80 CA12 (0.56) CYP11B1CYP11B2NAPRTNR1H3L3MBTL1
SCHEMBL10169507 0.78 HSD17B1 (0.48) HSD17B1HSD17B2NR1H3L3MBTL1
SCHEMBL18085884 0.77 LMNA (0.55) HSD17B1HSD17B2L3MBTL1
SCHEMBL10169508 0.77 FFAR1 (0.50) HSD17B1HSD17B2NR1H3L3MBTL1
SCHEMBL10169504 0.76 HSD17B1 (0.59) HSD17B1HSD17B2NR1H3L3MBTL1
SCHEMBL10169506 0.76 NPC1 (0.60) HSD17B1HSD17B2L3MBTL1
SCHEMBL10169213 0.74 ALDH1A1 (0.48) L3MBTL1
SCHEMBL5609778 0.73 CYP11B1 (0.49) CYP11B1CYP11B2HSD17B1HSD17B2NAPRT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8586751-B2 Nicotinamide compounds useful as kinase modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2013-11-19 US disclosed
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MEYERS SQUIBB COMPANY 2012-04-05 US disclosed
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MEYERS SQUIBB COMPANY 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120082702-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS NADK, BTK, NAMPT CYP11B1 1363/4885CYP11B2 1625/4885GRM2 2419/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.