SCHEMBL10172768

SCHEMBL10172768

CCOC(=O)C(C(=O)OC(C)(C)C)c1sc(Cl)cc1[N+](=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 3/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
MEN1 O00255 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
THRB P10828 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10160125 0.89 MAPT (0.39) KMT2ALMNAMAPTALDH1A1HPGD
SCHEMBL359022 0.69 THRB (0.43) KMT2ALMNAMAPTALDH1A1PKM
SCHEMBL10727958 0.67 CYP3A4 (0.47) KMT2ALMNAMAPTALDH1A1KDM4E
SCHEMBL16920141 0.67 ALDH1A1 (0.41) KMT2ALMNAMAPTALDH1A1L3MBTL1
SCHEMBL3961361 0.65 KMT2A (0.44) KMT2ALMNAMAPTALDH1A1L3MBTL1
SCHEMBL16522671 0.64 KMT2A (0.47) KMT2ALMNAMAPTALDH1A1KDM4E
SCHEMBL3968921 0.64 ALDH1A1 (0.39) KMT2ALMNAMAPTALDH1A1L3MBTL1
SCHEMBL27958738 0.64 MAPT (0.42) KMT2ALMNAMAPTALDH1A1KDM4E
SCHEMBL17083920 0.64 ALDH1A1 (0.64) KMT2ALMNAMAPTALDH1A1KDM4E
SCHEMBL16795576 0.64 MMP8 (0.60) KMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012022707-A1 SUBSTITUTED HETEROARYL SPIROPYRROLIDINE MDM2 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2012-02-23 WO disclosed