SCHEMBL10173167

SCHEMBL10173167

CCCNC(=O)CCNC(=O)CC

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58
CASP2 P42575 1/20 0.48
MCL1 Q07820 1/20 0.48
CNR1 P21554 1/20 0.46
NAAA Q02083 1/20 0.45
EPHX1 P07099 1/20 0.45
FAAH O00519 3/20 0.44
MMP1 P03956 1/20 0.41
MMP2 P08253 1/20 0.41
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
DNM1 Q05193 1/20 0.41
GAA P10253 1/20 0.41
CTSD P07339 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL165731 0.90
SCHEMBL11347096 0.87
SCHEMBL11334186 0.87
SCHEMBL11330562 0.87
SCHEMBL12673154 0.86 KMT2A (0.58) KMT2AMEN1CASP2MCL1NAAA
SCHEMBL3351989 0.85 CASP2 (0.56) KMT2AMEN1CASP2MCL1CNR1
SCHEMBL23728846 0.84 CASP2 (0.47) KMT2AMEN1CASP2MCL1CNR1
SCHEMBL12673157 0.83 CASP2 (0.61) KMT2AMEN1CASP2NAAAFAAH
SCHEMBL19544668 0.83 MEN1 (0.68) KMT2AMEN1CASP2CNR1NAAA
SCHEMBL30185947 0.82 EPHX1 (0.63) KMT2AMEN1CASP2NAAAEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020206137-A1 CDK2/5 DEGRADERS AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-10-08 WO disclosed
US-20150314008-A1 AURISTATIN COMPOUNDS AND CONJUGATES THEREOF MERSANA THERAPEUTICS, INC. 2015-11-05 US disclosed
US-20120022245-A1 FOLATE TARGETING OF NUCLEOTIDES PURDUE RESEARCH FOUNDATION (US) 2012-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120022245-A1 FOLATE TARGETING OF NUCLEOTIDES FOLR1, FOLR2, DHFR KMT2A 1861/4885MEN1 3080/4885CASP2 3941/4885
US-20150314008-A1 AURISTATIN COMPOUNDS AND CONJUGATES THEREOF PBRM1, BRWD1, BRDT KMT2A 1344/4885MEN1 2807/4885CASP2 3155/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.