SCHEMBL10175124

SCHEMBL10175124

Cn1c(-c2cncc(F)c2)nc2cc(Br)c(F)cc21

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 13/20 0.51
CYP11B1 P15538 12/20 0.51
CYP19A1 P11511 2/20 0.51
ADRA2B P18089 1/20 0.51
TLR7 Q9NYK1 3/20 0.39
ALOX15 P16050 1/20 0.36
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CYP3A4 P08684 1/20 0.34
PIM1 P11309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896599 0.89 CYP11B2 (0.63) CYP11B2CYP11B1CYP19A1ADRA2BALOX15
SCHEMBL10175129 0.87 CYP11B2 (0.45) CYP11B2CYP11B1CYP19A1ADRA2BALOX15
SCHEMBL17896646 0.85 CYP11B1 (0.57) CYP11B2CYP11B1CYP19A1ADRA2BCYP3A4
SCHEMBL17896771 0.84 CYP11B1 (0.54) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL17896647 0.82 CYP11B2 (0.67) CYP11B2CYP11B1HTTATM
SCHEMBL17896640 0.81 CYP11B2 (0.66) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL17896619 0.81 NPC1 (0.51) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL462213 0.81 CYP11B2 (0.55) CYP11B2CYP11B1CYP19A1ADRA2BALOX15
SCHEMBL10175145 0.81 CYP11B2 (0.55) CYP11B2CYP11B1CYP19A1ADRA2BALOX15
SCHEMBL17896718 0.79 CYP11B2 (0.56) CYP11B2CYP11B1CYP19A1ADRA2BATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed