SCHEMBL10175447

SCHEMBL10175447

Cn1c(-c2cccnc2)nc2ccc(F)c(F)c21

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 15/20 0.60
CYP11B1 P15538 9/20 0.60
DPP4 P27487 1/20 0.51
DPP8 Q6V1X1 1/20 0.51
ATM Q13315 1/20 0.43
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
CHRNB2 P17787 1/20 0.42
CHRNA5 P30532 1/20 0.42
CHRNA4 P43681 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175592 0.82 CYP11B2 (0.76) CYP11B2CYP11B1
SCHEMBL17896769 0.81 CYP11B2 (0.48) CYP11B2CYP11B1DPP4DPP8MAPT
SCHEMBL10176205 0.81 CYP11B2 (0.56) CYP11B2CYP11B1
SCHEMBL10175459 0.81 CYP11B2 (0.56) CYP11B2CYP11B1
SCHEMBL17896700 0.80 CYP11B2 (0.62) CYP11B2CYP11B1DPP4DPP8ATM
SCHEMBL17896705 0.78 CYP11B2 (0.54) CYP11B2CYP11B1DPP4DPP8
SCHEMBL463351 0.78 CYP11B2 (0.67) CYP11B2CYP11B1
SCHEMBL10175451 0.78 CYP11B2 (0.63) CYP11B2CYP11B1
SCHEMBL17897057 0.76 CYP11B2 (0.52) CYP11B2CYP11B1
SCHEMBL17896707 0.76 CYP11B2 (0.52) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed