SCHEMBL10175451

SCHEMBL10175451

Cc1cnccc1-c1nc2ccc(F)c(F)c2n1C

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.63
PDE10A Q9Y233 14/20 0.46
PDE2A O00408 12/20 0.43
PDE7A Q13946 2/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
PDE11A Q9HCR9 1/20 0.40
CYP11B1 P15538 2/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
S1PR1 P21453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL463351 0.89 CYP11B2 (0.67) CYP11B2PDE10APDE2APDE7ANOS2
SCHEMBL10175449 0.86 CYP11B2 (0.60) CYP11B2PDE10APDE2APDE7ANOS3
SCHEMBL10175463 0.83 CYP11B2 (0.67) CYP11B2PDE10ACYP11B1
SCHEMBL17896713 0.83 CYP11B2 (0.53) CYP11B2PDE10APDE2ACYP11B1
SCHEMBL10175118 0.83 CYP11B2 (0.57) CYP11B2PDE10ACYP11B1POLBSMN1; SMN2
SCHEMBL17896706 0.82 CYP11B2 (0.61) CYP11B2PDE10APDE2APDE7ACYP11B1
SCHEMBL17896708 0.79 CYP11B2 (0.68) CYP11B2CYP11B1
SCHEMBL10175447 0.78 CYP11B2 (0.60) CYP11B2CYP11B1
SCHEMBL10175445 0.77 CYP11B2 (1.00) CYP11B2CYP11B1
SCHEMBL17897047 0.74 CYP11B2 (0.61) CYP11B2PDE10APDE2ACYP11B1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed