SCHEMBL17896705

SCHEMBL17896705

Cn1c(-c2cncc(Br)c2)nc2ccc(F)c(F)c21

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 13/20 0.54
CYP11B1 P15538 9/20 0.41
PTGS2 P35354 2/20 0.41
CYP2A6 P11509 2/20 0.37
CYP19A1 P11511 3/20 0.34
ADRA2B P18089 2/20 0.34
ADRB1 P08588 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2C P18825 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
TLR7 Q9NYK1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175459 0.86 CYP11B2 (0.56) CYP11B2CYP11B1PTGS2CYP2A6CYP19A1
SCHEMBL10176205 0.86 CYP11B2 (0.56) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL17896709 0.83 CYP11B2 (0.61) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL17896707 0.82 CYP11B2 (0.52) CYP11B2CYP11B1PTGS2CYP19A1ADRA2B
SCHEMBL17897057 0.82 CYP11B2 (0.52) CYP11B2CYP11B1PTGS2
SCHEMBL10175455 0.81 CYP11B2 (0.51) CYP11B2CYP11B1TLR7
SCHEMBL17896699 0.80 PTGS2 (0.39) CYP11B2CYP11B1PTGS2CYP2A6CYP19A1
SCHEMBL10175447 0.78 CYP11B2 (0.60) CYP11B2CYP11B1DPP4DPP8
SCHEMBL10175145 0.77 CYP11B2 (0.55) CYP11B2CYP11B1PTGS2CYP19A1ADRA2B
SCHEMBL17896692 0.75 CYP11B1 (0.46) CYP11B2CYP11B1PTGS2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed