SCHEMBL10175602

SCHEMBL10175602

Cn1c(-c2cncc(C(F)(F)F)c2)nc2cc(C(F)(F)F)ccc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.51
HTR6 P50406 1/20 0.51
KIT P10721 2/20 0.49
CYP11B2 P19099 9/20 0.43
CYP11B1 P15538 6/20 0.43
CYP19A1 P11511 2/20 0.40
AGPAT2 O15120 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
ATM Q13315 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HTR2C P28335 2/20 0.39
ADRB1 P08588 1/20 0.39
ADRA2A P08913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896628 0.90 HTR2B (0.46) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL17896629 0.88 PTGS2 (0.49) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL17896627 0.86 PTGS2 (0.51) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL17883795 0.85 CYP11B2 (0.47) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL17896630 0.84 NPBWR1 (0.48) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL17896626 0.84 HTR2B (0.67) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL167098 0.83 MEN1 (0.57) HTR2BHTR6KITAGPAT2PIK3CA
SCHEMBL10175601 0.81 HTR2B (0.43) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL17883786 0.81 CYP11B2 (0.46) HTR2BKITCYP11B2CYP11B1CYP19A1
SCHEMBL17896614 0.78 CYP11B2 (0.49) HTR2BCYP11B2CYP11B1CYP19A1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed