SCHEMBL17896629

SCHEMBL17896629

Cn1c(-c2cncc(Br)c2)nc2cc(C(F)(F)F)ccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.49
HTR2B P41595 1/20 0.46
HTR6 P50406 1/20 0.46
KIT P10721 2/20 0.45
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP11B2 P19099 5/20 0.39
CYP11B1 P15538 4/20 0.39
PKM P14618 1/20 0.39
PDE2A O00408 1/20 0.38
AGPAT2 O15120 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175602 0.88 HTR2B (0.51) HTR2BHTR6KITTP53TSHR
SCHEMBL17896628 0.86 HTR2B (0.46) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL17896627 0.83 PTGS2 (0.51) PTGS2HTR2BHTR6KITCYP11B2
SCHEMBL17896634 0.81 HTR2B (0.71) HTR2BHTR6CYP11B2CYP11B1PKM
SCHEMBL17896630 0.81 NPBWR1 (0.48) HTR2BHTR6KITTP53TSHR
SCHEMBL17896626 0.81 HTR2B (0.67) PTGS2HTR2BHTR6KITCYP11B2
SCHEMBL167098 0.80 MEN1 (0.57) HTR2BHTR6KITNPC1ALDH1A1
SCHEMBL460705 0.79 ACSS2 (0.45) NPC1ALDH1A1TP53MAPTALOX15
SCHEMBL10175601 0.78 HTR2B (0.43) HTR2BHTR6KITCYP11B2CYP11B1
SCHEMBL10175145 0.78 CYP11B2 (0.55) PTGS2ALOX15CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed