SCHEMBL10175604

SCHEMBL10175604

CCOn1c(-c2cccnc2)nc2cc(SC)ccc21

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 13/20 0.43
CYP11B1 P15538 9/20 0.43
ALOX5AP P20292 1/20 0.40
USP2 O75604 1/20 0.39
HTT P42858 1/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
HTR2B P41595 1/20 0.38
HTR6 P50406 1/20 0.38
CYP19A1 P11511 1/20 0.38
DHFR P00374 1/20 0.37
RAD51 Q06609 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL458763 0.87 CYP11B2 (0.43) CYP11B2CYP11B1ALOX5APUSP2HTT
SCHEMBL17896749 0.84 CYP11B2 (0.45) CYP11B2CYP11B1ALOX5APUSP2HTT
SCHEMBL17896747 0.81 PTGS2 (0.46) CYP11B2CYP11B1ALOX5APUSP2HTT
SCHEMBL17896746 0.80 CYP11B2 (0.42) CYP11B2CYP11B1ALOX5APUSP2HTT
SCHEMBL458936 0.80 CYP11B2 (0.44) CYP11B2CYP11B1ALOX5APUSP2HTT
SCHEMBL10175792 0.70 CYP11B2 (0.46) CYP11B2CYP11B1ALOX5APUSP2HTT
SCHEMBL17896751 0.70 MAPT (0.49) CYP11B2CYP11B1CYP19A1LMNAPOLB
SCHEMBL17896748 0.68 USP2 (0.47) CYP11B2CYP11B1ALOX5APUSP2HTT
SCHEMBL459209 0.68 PTGS2 (0.48) CYP11B2CYP11B1ALOX5APUSP2HTT
SCHEMBL17896752 0.67 CYP11B1 (0.44) CYP11B2CYP11B1USP2HTTCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed