SCHEMBL458936

SCHEMBL458936

CSc1ccc2c(c1)nc(-c1cccnc1)n2O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 11/20 0.44
CYP11B1 P15538 9/20 0.44
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
ALOX5AP P20292 1/20 0.43
RAD51 Q06609 2/20 0.42
HTR2B P41595 1/20 0.41
HTR6 P50406 1/20 0.41
DHFR P00374 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL458763 0.82 CYP11B2 (0.43) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10175607 0.80 CYP11B2 (0.49) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10175604 0.80 CYP11B2 (0.43) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL17896745 0.79 PTGS2 (0.51) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL17896750 0.78 CYP11B2 (0.43) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL17897056 0.75 MET (0.49) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL17896753 0.72 CYP11B2 (0.50) CYP11B2CYP11B1KDM4EGAA
SCHEMBL12325780 0.68 RAB9A (0.54) CYP11B2CYP11B1ALDH1A1MAPT
SCHEMBL10176218 0.67 CYP11B2 (0.60) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10175606 0.67 CYP11B2 (0.60) CYP11B2CYP11B1USP2HTTNCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed