SCHEMBL10176202

SCHEMBL10176202

Cn1c(-c2cccnc2)nc2cc(F)c(F)cc21

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 13/20 0.73
CYP11B1 P15538 10/20 0.73
ATM Q13315 1/20 0.51
KIT P10721 3/20 0.48
USP2 O75604 1/20 0.47
HTT P42858 1/20 0.47
NCOA1 Q15788 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
NAMPT P43490 1/20 0.46
HTR2B P41595 1/20 0.44
HTR6 P50406 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896740 0.89 CYP11B2 (0.67) CYP11B2CYP11B1ATMKITUSP2
SCHEMBL17896647 0.89 CYP11B2 (0.67) CYP11B2CYP11B1ATMKITUSP2
SCHEMBL10176167 0.84 CYP11B2 (0.80) CYP11B2CYP11B1ATMKITUSP2
SCHEMBL10176164 0.84 CYP11B2 (1.00) CYP11B2CYP11B1ATMKITUSP2
SCHEMBL17896590 0.82 CYP11B2 (0.75) CYP11B2CYP11B1
SCHEMBL17896765 0.80 CYP11B2 (0.58) CYP11B2CYP11B1HTTHTR2BHTR6
SCHEMBL17896599 0.79 CYP11B2 (0.63) CYP11B2CYP11B1HTTHTR2B
SCHEMBL17883792 0.79 CYP11B2 (0.58) CYP11B2CYP11B1HTT
SCHEMBL1104859 0.79 MEN1 (0.69) CYP11B2CYP11B1ATMUSP2HTT
SCHEMBL10176218 0.79 CYP11B2 (0.60) CYP11B2CYP11B1ATMKITUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed