SCHEMBL10176218

SCHEMBL10176218

Cn1c(-c2cccnc2)nc2cc(N)ccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.60
CYP11B1 P15538 5/20 0.60
ATM Q13315 1/20 0.54
HTT P42858 3/20 0.53
KDM4E B2RXH2 2/20 0.53
NPC1 O15118 2/20 0.53
ALDH1A1 P00352 2/20 0.53
HSD17B10 Q99714 2/20 0.53
MAPT P10636 2/20 0.53
POLB P06746 1/20 0.53
HPGD P15428 1/20 0.53
GFER P55789 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
TP53 P04637 1/20 0.51
GAA P10253 1/20 0.51
PKM P14618 1/20 0.51
ALOX15 P16050 1/20 0.51
RAB9A P51151 1/20 0.51
ALOX5AP P20292 1/20 0.51
NAMPT P43490 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3158636 0.84 ALDH1A1 (0.67) ATMHTTKDM4ENPC1ALDH1A1
SCHEMBL10175606 0.83 CYP11B2 (0.60) CYP11B2CYP11B1ATMHTTNPC1
SCHEMBL10176167 0.83 CYP11B2 (0.80) CYP11B2CYP11B1ATMHTTALOX5AP
SCHEMBL1378639 0.83 CYP11B2 (0.62) CYP11B2CYP11B1HTTKDM4EALDH1A1
SCHEMBL20982514 0.82 KDM4E (0.68) ATMHTTKDM4ENPC1ALDH1A1
SCHEMBL10175817 0.81 RAD51 (0.60) CYP11B2CYP11B1ATMKDM4ENPC1
SCHEMBL1104859 0.81 MEN1 (0.69) CYP11B2CYP11B1ATMHTTKDM4E
SCHEMBL2251213 0.81 KDM4E (0.71) ATMHTTKDM4ENPC1ALDH1A1
SCHEMBL17883781 0.80 PTGS2 (0.57) CYP11B2CYP11B1ATMNPC1RAB9A
SCHEMBL17896626 0.80 HTR2B (0.67) CYP11B2CYP11B1ATMALOX5APNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed