SCHEMBL10176228

SCHEMBL10176228

CC(C)n1c(-c2cccnc2)nc2cc(Br)ccc21

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.70
HTT P42858 1/20 0.70
NCOA1 Q15788 1/20 0.70
NCOA3 Q9Y6Q9 1/20 0.70
CYP11B2 P19099 12/20 0.62
CYP11B1 P15538 10/20 0.62
ALOX5AP P20292 1/20 0.43
HTR2B P41595 1/20 0.41
HTR6 P50406 1/20 0.41
G6PD P11413 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
ALPG P10696 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
HSD17B10 Q99714 1/20 0.40
DHFR P00374 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175606 0.83 CYP11B2 (0.60) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL17896748 0.82 USP2 (0.47) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL10175131 0.81 USP2 (0.65) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL10175607 0.80 CYP11B2 (0.49) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL17896625 0.80 CYP11B2 (0.62) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL10175792 0.80 CYP11B2 (0.46) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL17883790 0.78 USP2 (0.63) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL10176165 0.77 CYP11B2 (1.00) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL17896749 0.77 CYP11B2 (0.45) USP2HTTNCOA1NCOA3CYP11B2
SCHEMBL10176229 0.76 CYP11B2 (0.74) CYP11B2CYP11B1HTR2BHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed