SCHEMBL10175607

SCHEMBL10175607

On1c(-c2cccnc2)nc2cc(Br)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 10/20 0.49
CYP11B1 P15538 8/20 0.49
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
ATM Q13315 1/20 0.46
RAD51 Q06609 1/20 0.44
HTR2B P41595 1/20 0.44
HTR6 P50406 1/20 0.44
RXFP1 Q9HBX9 2/20 0.43
G6PD P11413 1/20 0.43
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
ALOX5AP P20292 1/20 0.43
PRNP P04156 1/20 0.43
PPARG P37231 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NR2E3 Q9Y5X4 1/20 0.43
NCOR2 Q9Y618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896753 0.89 CYP11B2 (0.50) CYP11B2CYP11B1KMT2AMEN1ATM
SCHEMBL10175606 0.83 CYP11B2 (0.60) CYP11B2CYP11B1KMT2AMEN1ATM
SCHEMBL17896625 0.80 CYP11B2 (0.62) CYP11B2CYP11B1KMT2AMEN1USP2
SCHEMBL10175792 0.80 CYP11B2 (0.46) CYP11B2CYP11B1RAD51HTR2BHTR6
SCHEMBL458936 0.80 CYP11B2 (0.44) CYP11B2CYP11B1RAD51HTR2BHTR6
SCHEMBL10176228 0.80 USP2 (0.70) CYP11B2CYP11B1KMT2AHTR2BHTR6
SCHEMBL17896745 0.79 PTGS2 (0.51) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10176229 0.79 CYP11B2 (0.74) CYP11B2CYP11B1HTR2BHTR6
SCHEMBL17896750 0.78 CYP11B2 (0.43) CYP11B2CYP11B1RAD51HTR2BHTR6
SCHEMBL17896748 0.78 USP2 (0.47) CYP11B2CYP11B1KMT2ARAD51HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed