SCHEMBL10175606

SCHEMBL10175606

Cn1c(-c2cccnc2)nc2cc(Br)ccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 7/20 0.60
CYP11B1 P15538 6/20 0.60
ATM Q13315 1/20 0.54
NPC1 O15118 1/20 0.52
ALDH1A1 P00352 1/20 0.52
TP53 P04637 1/20 0.52
MAPT P10636 1/20 0.52
ALOX15 P16050 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
NAMPT P43490 1/20 0.51
USP2 O75604 1/20 0.46
HTT P42858 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
ALOX5AP P20292 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30663914 0.89 CYP11B2 (0.71) CYP11B2CYP11B1ATMUSP2HTT
SCHEMBL8209154 0.89 CYP11B2 (0.71) CYP11B2CYP11B1ATMUSP2HTT
SCHEMBL337983 0.84 ALDH1A1 (0.58) ATMNPC1ALDH1A1TP53MAPT
SCHEMBL10176167 0.83 CYP11B2 (0.80) CYP11B2CYP11B1ATMNAMPTUSP2
SCHEMBL10175607 0.83 CYP11B2 (0.49) CYP11B2CYP11B1ATMMAPTUSP2
SCHEMBL10176218 0.83 CYP11B2 (0.60) CYP11B2CYP11B1ATMNPC1ALDH1A1
SCHEMBL17896625 0.83 CYP11B2 (0.62) CYP11B2CYP11B1ALDH1A1MAPTTSHR
SCHEMBL10176228 0.83 USP2 (0.70) CYP11B2CYP11B1ALDH1A1TP53MAPT
SCHEMBL10175792 0.83 CYP11B2 (0.46) CYP11B2CYP11B1NPC1RAB9AUSP2
SCHEMBL17896623 0.82 MEN1 (0.62) ATMNPC1ALDH1A1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed