SCHEMBL1018019

SCHEMBL1018019

CC(C)(C)C(NC(=O)O)C1CCN(c2nc(Cl)ncc2-c2ccncc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.35
CNR2 P34972 1/20 0.35
HCRTR2 O43614 3/20 0.35
ABL1 P00519 2/20 0.35
BCR P11274 1/20 0.35
ROCK2 O75116 2/20 0.34
ROCK1 Q13464 2/20 0.34
CKS1B P61024 3/20 0.34
SKP1 P63208 3/20 0.34
SKP2 Q13309 3/20 0.34
CYP46A1 Q9Y6A2 1/20 0.33
SLC2A1 P11166 1/20 0.33
GPR6 P46095 1/20 0.33
NEK2 P51955 1/20 0.33
ADORA2B P29275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1018733 0.82 ABL1 (0.51) HCRTR2ABL1BCRCKS1BSKP1
SCHEMBL1018116 0.81 ABL1 (0.39) CNR2HCRTR2ABL1BCRCKS1B
SCHEMBL4304296 0.77 ROCK2 (0.44) ROCK2ROCK1CKS1BSKP1SKP2
SCHEMBL785864 0.77 ITGB3 (0.43) SLC2A1
SCHEMBL4304300 0.76 F10 (0.39) HCRTR2ABL1BCRROCK2ROCK1
SCHEMBL1018020 0.76 ROCK2 (0.37) HCRTR2ROCK2ROCK1CKS1BSKP1
SCHEMBL12082948 0.74 CKS1B (0.54) ROCK2ROCK1CKS1BSKP1SKP2
SCHEMBL1021391 0.74 RAF1 (0.32) ABL1BCRCKS1BSKP1SKP2
SCHEMBL27809364 0.74 AAK1 (0.44) HCRTR2ABL1BCRCYP46A1
SCHEMBL1938711 0.70 TSHR (0.55) NEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271631-A2 INHIBITORS OF PROTEIN KINASES Portola Pharmaceuticals, Inc. (US) 2011-01-12 EP disclosed
WO-2009131687-A2 INHIBITORS OF PROTEIN KINASES PORTOLA PHARMACEUTICALS, INC. (US) 2009-10-29 WO disclosed