SCHEMBL10180210

SCHEMBL10180210

CS(=O)(=O)c1ccc2c(c1)CCN2Cc1ccc(C2CCN(C(=O)O)CC2)cn1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 10/20 0.45
PRMT5 O14744 9/20 0.43
DRD3 P35462 1/20 0.39
HTR6 P50406 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10179692 0.95 GPR119 (0.41) GPR119PRMT5
SCHEMBL10179554 0.87 GPR119 (0.45) GPR119
SCHEMBL10179268 0.85 PRMT5 (0.41) GPR119PRMT5
SCHEMBL10179091 0.81 GPR119 (0.45) GPR119DRD3HTR6HRH3
SCHEMBL10179883 0.78 DRD2 (0.36) GPR119PRMT5HRH3
SCHEMBL10181085 0.78 CCR2 (0.38) GPR119PRMT5
SCHEMBL10180791 0.78 IRAK4 (0.37) GPR119PRMT5
SCHEMBL10179713 0.78 GPR119 (0.39) GPR119PRMT5
SCHEMBL10179608 0.77 THRA (0.35) GPR119PRMT5
SCHEMBL1577441 0.77 GPR119 (0.44) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2474540-A1 GPR119 AGONIST Nippon Chemiphar Co., Ltd. (JP) 2012-07-11 EP disclosed