SCHEMBL1018117

SCHEMBL1018117

CC(C)(C)N(CC1CCN(c2nc(Cl)ncc2C2CC2)CC1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.39
NEK2 P51955 1/20 0.33
PDE10A Q9Y233 7/20 0.33
HCRTR2 O43614 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32
ABL1 P00519 2/20 0.32
BCR P11274 2/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
SIRT3 Q9NTG7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1018735 0.86 ABL1 (0.46) HCRTR2SMN1; SMN2ABL1BCR
SCHEMBL1018020 0.81 ROCK2 (0.37) PDE10AHCRTR2CKS1BSKP1SKP2
SCHEMBL4307476 0.80 SMN1; SMN2 (0.36) NEK2HCRTR2SMN1; SMN2ABL1BCR
SCHEMBL1021392 0.78 ENPP1 (0.33) CKS1BSKP1SKP2SIRT2SIRT1
SCHEMBL4307471 0.77 CKS1B (0.41) CKS1BSKP1SKP2SIRT2SIRT1
SCHEMBL12083122 0.76 CKS1B (0.53) CKS1BSKP1SKP2SIRT2SIRT1
SCHEMBL27912561 0.75 PDE10A (0.44) CNR2PDE10AHCRTR2ABL1BCR
SCHEMBL1018116 0.73 ABL1 (0.39) CNR2NEK2HCRTR2SMN1; SMN2CKS1B
SCHEMBL343114 0.71 CRHR1 (0.33)
SCHEMBL2521770 0.70 PIM1 (0.36) CNR2NEK2SMN1; SMN2CKS1BSKP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271631-A2 INHIBITORS OF PROTEIN KINASES Portola Pharmaceuticals, Inc. (US) 2011-01-12 EP disclosed