SCHEMBL10188888

SCHEMBL10188888

Cc1cc(Cl)c(-c2nc3ccc(C#N)cc3[nH]2)cn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 1/20 0.51
PKN2 Q16513 1/20 0.51
METAP2 P50579 1/20 0.51
METAP1 P53582 1/20 0.51
RHEB Q15382 1/20 0.48
CSNK1D P48730 4/20 0.46
CSNK1A1 P48729 3/20 0.46
GSK3B P49841 3/20 0.46
CSNK1G2 P78368 3/20 0.46
KCNH2 Q12809 2/20 0.46
SSTR2 P30874 1/20 0.46
CHEK2 O96017 1/20 0.46
PIN1 Q13526 1/20 0.43
ATR Q13535 1/20 0.43
FASN P49327 1/20 0.42
DGAT1 O75907 1/20 0.41
SOAT1 P35610 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10188887 0.84 PKN1 (0.54) PKN1PKN2METAP2METAP1RHEB
SCHEMBL10189650 0.81 METAP2 (0.47) PKN1PKN2METAP2METAP1CSNK1D
SCHEMBL10188886 0.79 AMY1A (0.55) KDM4EALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL903006 0.79 METAP2 (0.61) PKN1PKN2METAP2METAP1CSNK1D
SCHEMBL10188890 0.77 SCD (0.58)
SCHEMBL20353609 0.76 PIN1 (0.47) PKN1PKN2METAP2METAP1RHEB
SCHEMBL1253278 0.74 PKN1 (0.58) PKN1PKN2METAP2METAP1RHEB
SCHEMBL902863 0.73 PKN1 (0.54) PKN1PKN2METAP2METAP1CSNK1D
SCHEMBL20982510 0.72 PKN1 (0.82) PKN1PKN2METAP2METAP1RHEB
SCHEMBL3341423 0.72 PKN1 (0.72) PKN1PKN2METAP2METAP1RHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed