SCHEMBL10195456

SCHEMBL10195456

O=C(c1ccc(-n2cc(-c3n[nH]c4c3=CCCC=4)nn2)cc1C(F)(F)F)N1CCOCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.37
EPHX2 P34913 2/20 0.35
RXRA P19793 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
LRRK2 Q5S007 7/20 0.34
NOTUM Q6P988 2/20 0.34
ABL1 P00519 2/20 0.34
BCR P11274 2/20 0.34
MAPK8 P45983 1/20 0.34
MAPK10 P53779 1/20 0.34
NTRK1 P04629 1/20 0.34
NTRK3 Q16288 1/20 0.34
NTRK2 Q16620 1/20 0.34
ALDH1A1 P00352 2/20 0.33
TSHR P16473 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194950 0.83 MAPK10 (0.44) GPR119LRRK2MAPK8MAPK10ALDH1A1
SCHEMBL22834181 0.74 GPR119 (0.41) GPR119RXRAGRIN1GRIN2BNOTUM
SCHEMBL10194693 0.72 LRRK2 (0.46) LRRK2MAPK8MAPK10ALDH1A1L3MBTL1
SCHEMBL10194888 0.72 MAPK10 (0.43) LRRK2MAPK8MAPK10ALDH1A1TSHR
SCHEMBL17850433 0.71 MAPK14 (0.36) LRRK2MAPK10
SCHEMBL17850412 0.69 ESRRA (0.48) GPR119RXRAGRIN1GRIN2BNOTUM
SCHEMBL10194754 0.69 JAK2 (0.47) EPHX2LRRK2MAPK8MAPK10
SCHEMBL10195054 0.69 MAPK1 (0.46) EPHX2MAPK8MAPK10
SCHEMBL22845788 0.69 P2RY14 (0.40) GPR119NOTUMTSHR
SCHEMBL29530740 0.69 P2RY14 (0.40) GPR119NOTUMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012084704-A1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO S.A. (CH) 2012-06-28 WO disclosed