SCHEMBL17850433

SCHEMBL17850433

O=C(c1ccc(-n2cc(-c3n[nH]c4c3=CCCC=4)nn2)cc1)N1CCOC(CO)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.36
ACKR3 P25106 1/20 0.36
LRRK2 Q5S007 2/20 0.34
ROCK2 O75116 1/20 0.34
JAK2 O60674 3/20 0.34
PIK3CA P42336 2/20 0.34
PIK3CD O00329 1/20 0.33
PIK3R2 O00459 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
PIK3R5 Q8WYR1 1/20 0.33
PIK3R3 Q92569 1/20 0.33
STAT3 P40763 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
LCK P06239 1/20 0.32
MGLL Q99685 1/20 0.31
DHODH Q02127 1/20 0.31
EGFR P00533 1/20 0.31
MAPK10 P53779 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194854 0.83 MAPK10 (0.42) MAPK14LRRK2ROCK2JAK2PIK3CA
SCHEMBL10194810 0.82 VNN1 (0.39) MAPK14JAK2MGLLEGFR
SCHEMBL10194707 0.77 MAPK10 (0.41) MAPK14ACKR3LRRK2ROCK2JAK2
SCHEMBL17850418 0.76 EGFR (0.36) MAPK14EGFRFLT3
SCHEMBL10194699 0.73 FLT3 (0.39) ACKR3LRRK2MAPK10FLT3
SCHEMBL10194859 0.72 FLT3 (0.42) LRRK2ROCK2JAK2PIK3CALCK
SCHEMBL10194868 0.72 ACKR3 (0.39) ACKR3JAK2
SCHEMBL10195456 0.71 GPR119 (0.37) LRRK2MAPK10
SCHEMBL10194993 0.70 FLT3 (0.46) LRRK2JAK2MAPK10FLT3
SCHEMBL10194775 0.68 FLT3 (0.44) LRRK2ROCK2JAK2LCKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed