SCHEMBL10197971

SCHEMBL10197971

Cn1cc(CP(C)(C)=O)c2c(Cl)cccc21

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.40
HTR2C P28335 5/20 0.40
HTR2B P41595 5/20 0.40
HTR2A P28223 4/20 0.39
P2RX7 Q99572 4/20 0.37
IL1B P01584 1/20 0.37
GPR84 Q9NQS5 1/20 0.37
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
KDR P35968 2/20 0.35
MCL1 Q07820 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
HTR6 P50406 2/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18508855 0.82 HTR2C (0.44) CDK2HTR2CHTR2BHTR2AGPR84
SCHEMBL8290971 0.82 HTR2C (0.39) CDK2HTR2CHTR2BHTR2AP2RX7
SCHEMBL3833273 0.76 CDK2 (0.47) CDK2HTR2CHTR2BHTR2AMCL1
SCHEMBL1093107 0.75 GPR84 (0.42) CDK2HTR2CHTR2BHTR2AP2RX7
SCHEMBL10197977 0.75 HTR2C (0.68) CDK2HTR2CHTR2BHTR2AGPR84
SCHEMBL10259878 0.75 HTR2A (0.41) CDK2HTR2CHTR2BHTR2AGPR84
Trimethylammonium SCHEMBL5399049 0.74 HTR2C (0.47) CDK2HTR2CHTR2BHTR2AGPR84
Iodide SCHEMBL5399054 0.74 CHRNB2 (0.41) CDK2HTR2CHTR2BHTR2AGPR84
SCHEMBL18509533 0.74 MCL1 (0.51) CDK2HTR2CHTR2BHTR2AMCL1
SCHEMBL14278470 0.73 SLC5A2 (0.43) CDK2HTR2CHTR2BHTR2AGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8546358-B2 Method of treating asthma JANSSEN PHARMACEUTICA NV (BE) 2013-10-01 US disclosed
US-20120022022-A1 NOVEL INHIBITORS OF CHYMASE HAWKINS MICHAEL J (US) 2012-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120022022-A1 NOVEL INHIBITORS OF CHYMASE CMA1, SERPINB1, TPSAB1 CDK2 827/4885HTR2C 3442/4885HTR2B 2346/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.