SCHEMBL1019865

SCHEMBL1019865

CS(=O)(=O)c1ccc(CNC(=O)c2cc(Cl)c[nH]c2=N)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CCR1 P32246 2/20 0.50
EPHX2 P34913 1/20 0.47
NR1H4 Q96RI1 1/20 0.47
TUBB P07437 2/20 0.46
MAPK8 P45983 3/20 0.44
MAPK9 P45984 3/20 0.44
CYP2C9 P11712 1/20 0.44
NAMPT P43490 1/20 0.44
KCNA5 P22460 1/20 0.44
MAPK10 P53779 2/20 0.44
PRKD3 O94806 1/20 0.44
MAPK1 P28482 1/20 0.44
PRKD2 Q9BZL6 1/20 0.44
ELANE P08246 2/20 0.43
NHERF1 O14745 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1019879 0.88 CCR1 (0.54) CCR1KCNA5ELANEALDH1A1GAA
SCHEMBL1016166 0.88 ALDH1A1 (0.50) CA1CA2CCR1TUBBNAMPT
SCHEMBL3487251 0.83 HSP90AA1 (0.52) CA1CA2TUBBKCNA5ADORA2A
SCHEMBL1017419 0.82 LMNA (0.44) CYP2C9ALDH1A1GAANPSR1
SCHEMBL1018589 0.80 DDR1 (0.48)
SCHEMBL15703882 0.80 EPHX2 (0.46) CA1CA2EPHX2KCNA5MAPK1
Hydrochloric Acid SCHEMBL1018259 0.79 DDR1 (0.47) EPHX2
Hydrochloric Acid SCHEMBL1016602 0.78 CCR1 (0.48) CCR1TUBBKCNA5MEN1KMT2A
SCHEMBL1017517 0.78 DDR1 (0.39) MAPK1ALDH1A1HSD17B10
SCHEMBL1016771 0.77 DDR1 (0.50) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271624-A1 IMINOPYRIDINE DERIVATIVES AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2011-01-12 EP claimed
WO-2009131245-A1 IMINOPYRIDINE DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-29 WO claimed
EP-2271624-A1 IMINOPYRIDINE DERIVATIVES AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2011-01-12 EP disclosed
WO-2009131245-A1 IMINOPYRIDINE DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-29 WO disclosed