SCHEMBL10208262

SCHEMBL10208262

CCOC(=O)c1ccc(-n2cc(N)c3cc(C(=O)N(C)Cc4ccccc4)ccc32)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.43
HTT P42858 2/20 0.42
RAB9A P51151 1/20 0.42
PPARG P37231 1/20 0.42
EGFR P00533 1/20 0.42
SRC P12931 1/20 0.42
KDR P35968 1/20 0.42
F2RL3 Q96RI0 1/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
POLB P06746 1/20 0.40
PRMT1 Q99873 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
BRPF1 P55201 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12309515 0.86 KDM4E (0.48)
SCHEMBL2736546 0.86 LMNA (0.44) HPGDALDH1A1MAPTHTTRAB9A
SCHEMBL2737111 0.85 MAPT (0.49) HPGDKMT2AALDH1A1MAPTHTT
SCHEMBL2736769 0.84 PTGER4 (0.41) HPGDALDH1A1MAPTHTTRAB9A
SCHEMBL10207671 0.81 EGFR (0.48) MEN1KMT2AMAPTHTTEGFR
SCHEMBL2736916 0.81 GABRA1 (0.46) MEN1KMT2ARAB9AEGFRSRC
SCHEMBL2736511 0.79 HPGD (0.47) HPGDKMT2AALDH1A1MAPTHTT
SCHEMBL2737105 0.78 CA12 (0.51) HPGDMEN1KMT2AALDH1A1MAPT
SCHEMBL12309620 0.74
SCHEMBL13594234 0.73 HDAC1 (0.48) ALDH1A1MAPTEGFRSRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402314-A1 (Aza)indole derivative and use thereof for medical purposes Kissei Pharmaceutical Co., Ltd. (JP) 2012-01-04 EP disclosed