SCHEMBL1022684

SCHEMBL1022684

COc1ccc([C@@H](C)CN)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.54
CA2 P00918 2/20 0.54
CA1 P00915 1/20 0.54
PPARG P37231 1/20 0.50
PPARD Q03181 1/20 0.50
PPARA Q07869 1/20 0.50
NFKB1 P19838 1/20 0.49
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ATM Q13315 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
ALOX12 P18054 1/20 0.47
TAAR1 Q96RJ0 2/20 0.45
KMT2A Q03164 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
CYP1A2 P05177 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29959275 1.00 ACHE (0.54) ACHECA2CA1PPARGPPARD
SCHEMBL1024752 1.00 ACHE (0.54) ACHECA2CA1PPARGPPARD
SCHEMBL3654988 1.00 ACHE (0.54) ACHECA2CA1PPARGPPARD
Bromide SCHEMBL11627374 0.98 ACHE (0.53) ACHECA2CA1PPARGPPARD
Bromide SCHEMBL11628156 0.98 ACHE (0.53) ACHECA2CA1PPARGPPARD
Bromide SCHEMBL11624070 0.98 ACHE (0.53) ACHECA2CA1PPARGPPARD
SCHEMBL20969576 0.85 SLC6A2 (0.43) ACHECA2CA1NFKB1BLM
SCHEMBL10843568 0.85 ACHE (0.51) ACHECA2CA1PPARGPPARD
SCHEMBL8298141 0.84 ALDH1A1 (0.60) ACHECA2CA1PPARGPPARD
SCHEMBL20969582 0.84 ADRA2A (0.46) ACHECA2CA1NFKB1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011000915-A1 ISOFORM-SELECTIVE HCN BLOCKERS UNIVERSITA' DEGLI STUDI DI FIRENZE (IT) 2011-01-06 WO disclosed
US-4581172-A Substituted pyrimido[6,1-a]isoquinolin-4-ones,pyrimido[6,1-a]benzozepin-4-ones and pyrimido[6,1-a]benzodiazepin-4-ones useful for prevention of thromboses and treating hypertension HOFFMANN-LA ROCHE INC. (US) 1986-04-08 US disclosed
US-4129580-A Resolution of certain asymmetric primary amines using lasalocid HOFFMANN-LA ROCHE INC. (US) 1978-12-12 US disclosed