SCHEMBL10238797

SCHEMBL10238797

Cc1cnc2c(c1)C(C)CC2

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
PDK2 Q15119 1/20 0.32
PDK4 Q16654 1/20 0.32
UGT2B17 O75795 2/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16692275 0.89 DRD2 (0.38) DRD2DRD1CA1CA2CCR1
SCHEMBL19985086 0.81 CA1 (0.36) CA1CA2
SCHEMBL21097488 0.79 DRD2 (0.39) DRD2DRD1CCR1CCR5CCR8
SCHEMBL24326944 0.77 PDPK1 (0.40) DRD2DRD1PDK2PDK4
SCHEMBL24336496 0.77 DRD2 (0.37) DRD2DRD1PDK2PDK4
SCHEMBL24336051 0.75 CA1 (0.39) CA1CA2
SCHEMBL20840970 0.73 DRD2 (0.37) DRD2DRD1NOS3NOS1NOS2
SCHEMBL10376879 0.73 DRD2 (0.37) DRD2DRD1PDK2PDK4UGT2B17
SCHEMBL31569169 0.73 MAOA (0.41) DRD2DRD1CYP2D6
SCHEMBL26571108 0.73 DRD2 (0.37) DRD2DRD1PDK2PDK4UGT2B17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8501804-B2 Bicyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-06 US disclosed
US-8501804-B2 Bicyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-06 US disclosed
US-20120010247-A1 BICYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-01-12 US disclosed
US-20120010247-A1 BICYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010247-A1 BICYCLIC COMPOUND ACACA, CPT1B, ACACB DRD2 4882/4885DRD1 4869/4885CA1 3637/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.