SCHEMBL1023948

SCHEMBL1023948

CC(=O)N(Cc1cccc(Nc2nc(Cl)ncc2Cl)c1)Cc1cccc(N(C(=O)OC(=O)C(F)(F)F)C(C)(C)C)c1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSC P53634 8/20 0.35
BCL6 P41182 1/20 0.35
BTK Q06187 3/20 0.33
EGFR P00533 4/20 0.33
MET P08581 2/20 0.32
PTK2 Q05397 2/20 0.32
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32
ITK Q08881 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1023947 0.88 CTSC (0.38) CTSCBCL6BTKEGFRMET
SCHEMBL4348211 0.86 BTK (0.38) CTSCBTKEGFRJAK3
SCHEMBL1026533 0.80 HSD11B1 (0.33)
Trifluoroacetic Acid SCHEMBL4348204 0.80 CTSC (0.41) CTSCBCL6BTKEGFRJAK3
SCHEMBL13623196 0.78 SYK (0.45) CTSCBCL6BTKEGFRMET
SCHEMBL1026395 0.77 BCL6 (0.40) CTSCBCL6BTKEGFRMET
SCHEMBL1026721 0.74 JAK3 (0.42) CTSCBCL6PTK2JAK2JAK3
SCHEMBL1023285 0.73 ALK (0.40) BCL6BTKMET
SCHEMBL1025086 0.72 BCL6 (0.38) CTSCBCL6BTKEGFRMET
SCHEMBL1026953 0.72 GAA (0.47) BCL6BTKMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274288-A2 MACROCYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS Incyte Corporation (US) 2011-01-19 EP disclosed